Cyclazocine meaning

Cyclazocine is a drug that acts as a κ-opioid receptor agonist and μ-opioid receptor antagonist.


Cyclazocine definitions

Word backwards enicozalcyc
Part of speech The word "cyclazocine" is a noun.
Syllabic division cy-cla-zo-cine
Plural The plural of cyclazocine is cyclazocines.
Total letters 11
Vogais (4) a,o,i,e
Consonants (5) c,y,l,z,n

Cyclazocine, a mixed agonist-antagonist drug, is classified as a kappa-opioid receptor agonist. Originally developed in the 1960s, it was intended for the treatment of pain but was later found to have potential for abuse due to its psychomimetic effects.

Chemical Properties

The chemical structure of cyclazocine includes a benzomorphan scaffold, making it a morphinan-type compound. It exhibits high affinity for the kappa-opioid receptor, which differentiates it from traditional opioids that primarily target mu-opioid receptors.

Uses

Cyclazocine is not approved for medical use in many countries due to its potential for abuse and addictive properties. However, it has been studied for its effects on mood, cognition, and behavior in various research settings. Some studies have explored its potential in treating depression and anxiety disorders.

Side Effects

Common side effects of cyclazocine may include dizziness, nausea, vomiting, constipation, and respiratory depression. Due to its interaction with the opioid receptors in the central nervous system, it can also lead to dependence and withdrawal symptoms if used improperly.

Despite its potential therapeutic benefits, the abuse liability of cyclazocine has limited its clinical use. It is considered a controlled substance in many countries, and its use is closely monitored. Research continues to investigate its pharmacological profile and potential applications in the field of neuropsychiatric disorders.


Cyclazocine Examples

  1. The doctor prescribed cyclazocine for the patient's severe pain.
  2. Researchers are studying the effects of cyclazocine on opioid receptors.
  3. Cyclazocine is a synthetic opioid analgesic used to treat moderate to severe pain.
  4. The pharmacokinetics of cyclazocine have been well-studied in clinical trials.
  5. Patients should not take cyclazocine with alcohol or other central nervous system depressants.
  6. Cyclazocine may cause side effects such as constipation, dizziness, and nausea.
  7. Individuals with a history of substance abuse should use cyclazocine with caution.
  8. Doctors should monitor patients closely for signs of respiratory depression when prescribing cyclazocine.
  9. It is important to follow the prescribed dosage of cyclazocine to avoid overdose.
  10. Cyclazocine should be stored in a secure place away from children and pets.


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  • Updated 21/06/2024 - 04:22:18